| A First-in-Human Phase 1 Study of a Novel Selective Androgen Receptor Modulator (SARM), RAD140, in ER+/HER2- Metastatic Breast Cancer.Clin Breast Cancer | No random groups | 2022 |
| Spontaneous Splenic Rupture in a Patient With Recent Use of Performance-Enhancing Compounds: A Case Report and Literature Review.Cureus | Case reports | 2026 |
| Cholestatic Drug-Induced Liver Injury From Rad-140 Successfully Treated With Corticosteroids.ACG Case Rep J | Case reports | 2025 |
| Selective Androgen Receptor Modulators Leading to Liver Injury: A Case Report.Cureus | Case reports | 2024 |
| Reversible Gynecomastia and Hypogonadism Due to Usage of Commercial Performance-Enhancing Supplement Use.JCEM Case Rep | Case reports | 2024 |
| Selective androgen receptor modulator abuse-induced heart failure: catastrophic effects of RAD-140 (Testolone).Pol Arch Intern Med | Case reports | 2024 |
| Myopericarditis Following Use of Selective Androgen Receptor Modifier "RAD-140".JACC Case Rep | Case reports | 2024 |
| Severe liver injury following use of RAD-140, a selective androgen receptor modulator, for body building.Aust Prescr | Case reports | 2024 |
| Idiosyncratic drug-induced liver injury related to use of novel selective androgen receptor modulator RAD140 (Testalone): a case report.J Med Case Rep | Case reports | 2023 |
| Selective Androgen Receptor Modulators (SARMs)-Induced Liver Injury: A Case Report and Review of Literature.Cureus | Case reports | 2023 |
| Acute Myocarditis From the Use of Selective Androgen Receptor Modulator (SARM) RAD-140 (Testolone).Cureus | Case reports | 2022 |
| Drug-Induced Liver Injury Associated With Alpha Bolic (RAD-140) and Alpha Elite (RAD-140 and LGD-4033).ACG Case Rep J | Case reports | 2020 |
| Detection of SARMs in doping control analysis.Mol Cell Endocrinol | Review of studies | 2018 |
| Treatment with a selective androgen receptor modulator (RAD140) is linked to better cardiac function, with male-specific effects that are graded by interleukin-6.Geroscience | In animals | 2026 |
| The impact of a selective androgen receptor modulator (RAD140) on frailty and underlying mechanisms in older male and female C57Bl/6 mice.Mech Ageing Dev | In animals | 2025 |
| Detection of nonsteroidal and steroidal selective androgen receptor modulators in equine hair after oral administrations.Drug Test Anal | In animals | 2025 |
| Identification of equine in vitro metabolites of seven non-steroidal selective androgen receptor modulators for doping control purposes.Drug Test Anal | In animals | 2022 |
| Label-free proteomics for discovering biomarker candidates of RAD140 administration to castrated horses.Drug Test Anal | In animals | 2021 |
| Metabolic studies of selective androgen receptor modulators RAD140 and S-23 in horses.Drug Test Anal | In animals | 2021 |
| Development of a multi-residue high-throughput UHPLC-MS/MS method for routine monitoring of SARM compounds in equine and bovine blood.Drug Test Anal | In animals | 2020 |
| Selective androgen receptor modulator RAD140 is neuroprotective in cultured neurons and kainate-lesioned male rats.Endocrinology | In animals | 2014 |
| Unregulated gains: a case of RAD-140-induced liver injury.Proc (Bayl Univ Med Cent) | Other paper | 2026 |
| Initial testing procedure based on microextraction followed by LC-HRMS analysis to determine 107 xenobiotics and their metabolites in serum/plasma.Analyst | Other paper | 2026 |
| Exploring transdermal SARMs exposure: analysis of the elimination profiles and metabolism for doping control purposes.J Anal Toxicol | Other paper | 2025 |
| Rapid detection of illegal selective androgen receptor modulators in unregistered supplements using a combination of selected solid-state analytical methods.ADMET DMPK | Other paper | 2025 |
| Deep Learning-Based Drug Compounds Discovery for Gynecomastia.Biomedicines | Other paper | 2025 |
| Detection of anabolic agents including selective androgen receptor modulators in samples outside of sport.Drug Test Anal | Other paper | 2024 |
| Social Interest Data as a Proxy for Off-Label Performance-Enhancing Drug Use: Implications and Clinical Considerations.Cureus | Other paper | 2024 |
| A rapid synthesis of molecularly imprinted polymer nanoparticles for the extraction of performance enhancing drugs (PIEDs).Nanoscale Adv | Other paper | 2023 |
| Comparison of in vitro approaches for predicting the metabolism of the selective androgen receptor modulator RAD140.Anal Bioanal Chem | Other paper | 2023 |
| Pharmacological Targeting of Androgen Receptor Elicits Context-Specific Effects in Estrogen Receptor-Positive Breast Cancer.Cancer Res | Other paper | 2023 |
| Detection of selective androgen receptor modulators (SARMs) in serum using a molecularly imprinted nanoparticle surface plasmon resonance sensor.J Mater Chem B | Other paper | 2022 |
| Human In Vivo Metabolism and Elimination Behavior of Micro-Dosed Selective Androgen Receptor Modulator RAD140 for Doping Control Purposes.Metabolites | Other paper | 2022 |
| Systematic identification of ACE2 expression modulators reveals cardiomyopathy as a risk factor for mortality in COVID-19 patients.Genome Biol | Other paper | 2022 |
| The forensic response after an adverse analytical finding (doping) involving a selective androgen receptor modulator (SARM) in human athlete.J Pharm Biomed Anal | Other paper | 2022 |
| Simultaneous detection of different chemical classes of selective androgen receptor modulators in urine by liquid chromatography-mass spectrometry-based techniques.J Pharm Biomed Anal | Other paper | 2021 |
| Comparison of the three SARMs RAD-140, GLPG0492 and GSK-2881078 in two different in vitro bioassays, and in an in silico androgen receptor binding assay.J Steroid Biochem Mol Biol | Other paper | 2019 |
| Selective Androgen Receptor Modulator RAD140 Inhibits the Growth of Androgen/Estrogen Receptor-Positive Breast Cancer Models with a Distinct Mechanism of Action.Clin Cancer Res | Other paper | 2017 |
| Expanding sports drug testing assays: mass spectrometric characterization of the selective androgen receptor modulator drug candidates RAD140 and ACP-105.Rapid Commun Mass Spectrom | Other paper | 2013 |
| Design, Synthesis, and Preclinical Characterization of the Selective Androgen Receptor Modulator (SARM) RAD140.ACS Med Chem Lett | Other paper | 2011 |